- Author:
Jinqin CHEN
1
;
Xinhong LIU
2
;
Shuo YU
1
;
Jia LIU
1
;
Rongfang CHEN
1
;
Yunxiao ZHANG
3
;
Ling JIANG
2
;
Qiuyun DAI
1
Author Information
- Publication Type:Journal Article
- Keywords: Analgesic activity; Bu8; DIEA, diisopropylethylamine; ESI-MS, electrospray ionization-mass spectroscopy; Fmoc, N-(9-fluorenyl)methyloxy-carbonyl; HBTU, 2-(1H-benzotriazol-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate; HOBt, 1-hydroxybenzotriazole; IC50, half-maximal inhibitory concentration; N-type calcium ion channel; RP-HPLC, reversed phase high-performance liquid chromatography; Structure–activity relationship; TFA, trifluoroacetic acid; ω-conotoxin
- From: Acta Pharmaceutica Sinica B 2021;11(9):2685-2693
- CountryChina
- Language:English