Mechanisms of resistance to crizotinib in patients with transforming EML4-ALK fusion gene.
10.3760/cma.j.issn.0529-5807.2012.12.020
- Author:
Hui-juan ZHANG
;
Xiao-tong ZHANG
;
Li ZHANG
- Publication Type:Journal Article
- MeSH:
Apoptosis;
drug effects;
Benzoquinones;
pharmacology;
Carcinoma, Non-Small-Cell Lung;
drug therapy;
metabolism;
pathology;
Drug Resistance, Neoplasm;
HSP90 Heat-Shock Proteins;
antagonists & inhibitors;
Humans;
Lactams, Macrocyclic;
pharmacology;
Lung Neoplasms;
drug therapy;
metabolism;
pathology;
Mutation;
Oncogene Proteins, Fusion;
antagonists & inhibitors;
genetics;
metabolism;
Protein Kinase Inhibitors;
therapeutic use;
Pyrazoles;
therapeutic use;
Pyridines;
therapeutic use;
Triazoles;
pharmacology
- From:
Chinese Journal of Pathology
2012;41(12):862-864
- CountryChina
- Language:Chinese